MedChemexpress LLC

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  • Company Name: MedChemexpress LLC
  • Street: 18 Wilkinson Way, Princeton, NJ 08540, USA
  • City: Princeton
  • Country/region: United States
  • Contact Person: Ms.James Gao
  • Tel: 609-228-6898
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CC-930

    Detailed Description

    CC-930CC-930(Tanzisertib) is a selective and potent JNK1/JNK2/JNK3(IC50=61/7/6 nM) inhibitor and is currently under clinical development for fibrotic and infammatory indications.

    IC50 Value: 61 nM (JNK1); 7 nM (JNK2); 6 nM (JNK3) [1]

    Target: JNK1/2/3

    in vitro: Compound 1 (CC-930) showed remarkable selectivity in a panel of 240 kinases, EGFR being the only non-MAP kinase inhibited more than 50% at 3 lM (IC50 = 0.38 lM).

    Target:/products

    Product Links:http://www.medchemexpress.cn/cc-930.html

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